Brevetti EPO No.3655395 2021.12.01
Brevetti EPO
(10) Registration Number and Date
2022000088 2022.02.23
Status
Expired
(180) Expiration Date
(20) Filing Number and Date
SM /T/2022/000088 2018.07.19
(40) Publication Number and Date
SM /T/2022/000088 2022.02.23
(30) Priority Details
US 201762534908 P
2017.07.20
(71/73) Applicant
(72) Inventor
(IT) CHAN, Collin : , New Brunswick, New Jersey 08903, US
(IT) FOREST, Robert V. : , New Brunswick, New Jersey 08903, US
(IT) RAZLER, Thomas M. : , New Brunswick, New Jersey 08903, US
(IT) EASTGATE, Martin D. : , New Brunswick, New Jersey 08903, US
(IT) LEE, Hong Geun : , Seoul 08826, KR
(IT) SAVAGE, Scott A. : , New Brunswick, New Jersey 08903, US
(IT) SFOUGGATAKIS, Chris : , New Brunswick, New Jersey 08903, US
(IT) FENSTER, Michael David Bengt : , New Brunswick, New Jersey 08903, US
(IT) LUO, Helen Y. : , San Francisco, CA 94117, US
(IT) GREEN, Rebecca A. : , New Brunswick, New Jersey 08903, US
(IT) LAUSER, Kathleen : , Minneapolis, MN 55414, US
(IT) DOMAGALSKI, Nathan R. : , Niantic, Connecticut 0637, US
(IT) GONZALEZ-BOBES, Francisco : , New Brunswick, New Jersey 08903, US
(IT) LA CRUZ, Thomas E. : , New Brunswick, New Jersey 08903, US
(IT) ZARETSKY, Serge : , New Brunswick, New Jersey 08903, US
(IT) AYTAR, Burcu Selin : , New Brunswick, New Jersey 08903, US
(IT) FAN, Yu : , Highland Park, NJ 08904, US
(IT) ZHU, Ye : , Singapore 129792, SG
(IT) KOPP, Nathaniel David : , New Brunswick, New Jersey 08903, US
(IT) LEAHY, David K. : , Marblehead, MA 01945, US
(IT) SOUMEILLANT, Maxime C.D. : , New Brunswick, New Jersey 08903, US
(74) Representative Name
(IT) SANTORO, Tiziana : Via 28 Luglio, 187, 47893 Borgo Maggiore RSM, SM
(54) Title
(IT) PROCEDIMENTO PER LA PREPARAZIONE DI N-((1R,2S,SR)-5-(TERT-BUTILAMMINO)-2-((S)-3-(7-TERT-BUTILPIRAZOLO[1,5-A][1,3,5]TRIAZIN-4-ILAMMINO)-2-OSSOPIRROLIDIN-1-IL)CICLOESIL)ACETAMMIDE
(EN) PROCESS FOR THE PREPARATION OF N-((1R,2S,SR)-5-(TERT-BUTYLAMINO)-2-((S)-3-(7-TERT-BUTYLPYRAZOLO[1,5-A][1,3,5]TRIAZIN-4-YLAMINO)-2-OXOPYRROLIDIN-1-YL)CYCLOHEXYL)ACETAMIDE
(57) Abstract
(58) Citations